SCHEMBL8935826

SCHEMBL8935826

COc1cccc(-c2cc(-c3cccc(CN(CC(=O)O)CC(=O)O)n3)nc(-c3cccc(CN(CC(=O)O)CC(=O)O)n3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
LTB4R Q15722 2/20 0.45
AVPR1B P47901 1/20 0.42
PTGER2 P43116 1/20 0.42
RECQL P46063 1/20 0.41
GRK6 P43250 1/20 0.41
HSD17B2 P37059 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
FFAR1 O14842 2/20 0.40
MAPK1 P28482 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
MAPT P10636 1/20 0.40
DHODH Q02127 1/20 0.40
BACE1 P56817 1/20 0.40
PIN1 Q13526 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765283 0.90 MCL1 (0.45) ADORA3LTB4RAVPR1BALDH1A1KDM4E
SCHEMBL13217240 0.87 MCL1 (0.42) ADORA3LTB4RAVPR1BALDH1A1KDM4E
SCHEMBL8601997 0.85 ALDH1A1 (0.44) ADORA3ALDH1A1KDM4EMAPK1MAPT
SCHEMBL8596932 0.85 MCL1 (0.41) ADORA3LTB4RAVPR1BALDH1A1KDM4E
SCHEMBL13997749 0.84 LTB4R (0.39) ADORA3ADORA2BADORA1LTB4RPTGER2
SCHEMBL8597039 0.83 MEN1 (0.44) ADORA3ADORA1LTB4RPTGER2KDM4E
SCHEMBL7717266 0.83 ADORA2A (0.37) ADORA3ALDH1A1KDM4E
SCHEMBL8935770 0.83 ALDH1A1 (0.42) ADORA3ALDH1A1KDM4EMAPK1
SCHEMBL9594479 0.82 MCL1 (0.37) LTB4RALDH1A1KDM4EMAPT
SCHEMBL8936038 0.82 ADORA2A (0.37) ADORA3ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539117-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines GE HEALTHCARE AS (NO) 1996-07-23 US disclosed
US-5350696-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines STERLING WINTHROP, INC. (US) 1994-09-27 US disclosed