SCHEMBL8935770

SCHEMBL8935770

COc1cc(-c2cc(-c3cccc(CN(CC(=O)O)CC(=O)O)n3)nc(-c3cccc(CN(CC(=O)O)CC(=O)O)n3)c2)ccc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MAPK1 P28482 1/20 0.37
PIK3CA P42336 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
GYS1 P13807 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
CHEK1 O14757 4/20 0.35
GAK O14976 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7717266 0.92 ADORA2A (0.37) ALDH1A1TSHRGYS1MEN1KMT2A
SCHEMBL30803820 0.92 ADORA2A (0.37) ALDH1A1TSHRGYS1MEN1KMT2A
SCHEMBL8936038 0.91 ADORA2A (0.37) ALDH1A1TSHRGYS1MEN1KMT2A
SCHEMBL8601997 0.90 ALDH1A1 (0.44) ALDH1A1TSHRHSD17B10MAPK1GYS1
SCHEMBL8935948 0.90 ADORA2A (0.36) ALDH1A1TSHRGYS1MEN1KMT2A
SCHEMBL7770333 0.86 ADORA2A (0.44) ALDH1A1TDP1MEN1KMT2AADORA2A
SCHEMBL8765283 0.84 MCL1 (0.45) ALDH1A1TSHRMAPK1GYS1ADORA3
SCHEMBL8935826 0.83 ADORA3 (0.46) ALDH1A1MAPK1ADORA3KDM4E
SCHEMBL13997750 0.82 LTB4R (0.41) ALDH1A1MEN1KMT2AKDM4EGAA
SCHEMBL9594349 0.82 LTB4R (0.41) ALDH1A1MEN1KMT2AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539117-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines GE HEALTHCARE AS (NO) 1996-07-23 US disclosed
US-5350696-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines STERLING WINTHROP, INC. (US) 1994-09-27 US disclosed