SCHEMBL8936165

SCHEMBL8936165

COc1cc(CBr)c2ccc(Cl)cc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.42
KDM4E B2RXH2 3/20 0.41
NR4A2 P43354 1/20 0.41
ELANE P08246 1/20 0.39
CHRM2 P08172 2/20 0.38
ADRA2C P18825 2/20 0.38
CHRM3 P20309 2/20 0.38
SLC6A2 P23975 2/20 0.38
DRD3 P35462 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 2/20 0.38
USP2 O75604 2/20 0.38
TP53 P04637 2/20 0.38
CYP3A4 P08684 2/20 0.38
CASP1 P29466 2/20 0.38
CASP7 P55210 2/20 0.38
HBB P68871 2/20 0.38
HSD17B10 Q99714 2/20 0.38
HTR1A P08908 2/20 0.38
ACHE P22303 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2190816 0.81 POLB (0.45) POLBKDM4ENR4A2ELANEACHE
SCHEMBL5639914 0.80 POLB (0.47) POLBKDM4ENR4A2ELANEACHE
SCHEMBL6629242 0.79 POLB (0.47) POLBKDM4EELANENPC1RAB9A
SCHEMBL8936095 0.79 POLB (0.64) POLBKDM4ENR4A2ELANEHSD17B10
SCHEMBL2419272 0.78 POLB (0.44) POLBNR4A2ACHECHRM1CYP1A2
SCHEMBL2417822 0.76 POLB (0.42) POLBKDM4ENR4A2USP2CYP3A4
SCHEMBL31590887 0.76 POLB (0.42) POLBKDM4ENR4A2USP2CYP3A4
SCHEMBL8936122 0.76 KDM4E (0.38) POLBKDM4ENR4A2ELANETP53
SCHEMBL3950903 0.73 NOS1 (0.32)
SCHEMBL23564604 0.70 ELANE (0.45) POLBKDM4ENR4A2ELANECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510338-A ADMINISTERING TO A MAMMAL TO RELIEVE PAIN AND TO TREAT CONVULSIONS, CEREBRAL ISCHEMIC DAMAGE, AND EMESIS GUILFORD PHARMACEUTICALS INC. (US) 1996-04-23 US disclosed
US-5342946-A Phosphonoalkylquinolin-2-ones as novel antagonists of non-NMDA ionotropic excitatory amino acid receptors GUILFORD PHARMACEUTICALS INC. (US) 1994-08-30 US disclosed