SCHEMBL8936508

SCHEMBL8936508

COc1ccccc1-c1c(NC(=O)NCc2ccccc2)n(C)c(=O)c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.59
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 2/20 0.51
ADORA3 P0DMS8 2/20 0.46
BRD4 O60885 1/20 0.46
HPGD P15428 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TP53 P04637 2/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
POLB P06746 1/20 0.44
PTPN1 P18031 1/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
SHMT2 P34897 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9178243 0.84 KDM4E (0.50) TACR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8936601 0.81 TACR1 (0.70) TACR1KDM4EALDH1A1ADORA3HPGD
SCHEMBL9179860 0.78 RAB9A (0.50) KDM4EALDH1A1BRD4HPGDNPSR1
SCHEMBL9177055 0.74 TACR1 (0.56) TACR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8936576 0.74 TACR1 (1.00) TACR1KDM4EALDH1A1ADORA3HPGD
SCHEMBL8936446 0.74 TACR1 (0.49) TACR1KDM4EALDH1A1TP53
SCHEMBL8936577 0.74 TACR1 (0.76) TACR1ALDH1A1TP53
SCHEMBL8784961 0.73 TACR1 (0.86) TACR1ALDH1A1HPGDTP53GAA
SCHEMBL8936431 0.73 TACR1 (0.56) TACR1KDM4EALDH1A1TP53
SCHEMBL8936535 0.73 TACR1 (0.73) TACR1ALDH1A1ADORA3HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5523305-A ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-04 US disclosed
EP-0566069-A1 Tachykinin receptor antagonists, isoquinolones and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-20 EP disclosed