SCHEMBL8936601

SCHEMBL8936601

Cn1c(NC(=O)NCc2ccccc2)c(-c2ccc(F)cc2)c2ccccc2c1=O

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.70
SMN1; SMN2 Q16637 3/20 0.50
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 2/20 0.50
LMNA P02545 2/20 0.50
HPGD P15428 1/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
MAOB P27338 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.45
USP2 O75604 1/20 0.45
MEN1 O00255 1/20 0.45
ADORA3 P0DMS8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936542 0.91 TACR1 (0.86) TACR1SMN1; SMN2ALDH1A1KDM4ELMNA
SCHEMBL8936429 0.89 TACR1 (0.61) TACR1SMN1; SMN2ALDH1A1KDM4ELMNA
SCHEMBL8936576 0.82 TACR1 (1.00) TACR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL8936577 0.82 TACR1 (0.76) TACR1ALDH1A1KMT2AMEN1
SCHEMBL8936508 0.81 TACR1 (0.59) TACR1ALDH1A1KDM4EHPGDPOLB
SCHEMBL9178393 0.79 TACR1 (0.57) TACR1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL8936527 0.78 TACR1 (0.90) TACR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL8936587 0.76 TACR1 (0.64) TACR1ALDH1A1KMT2AMEN1ADORA3
SCHEMBL8936439 0.76 TACR1 (0.86) TACR1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL8936454 0.76 TACR1 (0.86) TACR1ALDH1A1NPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5523305-A ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-04 US disclosed
EP-0566069-A1 Tachykinin receptor antagonists, isoquinolones and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-20 EP disclosed