SCHEMBL8936701

SCHEMBL8936701

CCNc1cc(Oc2ccc(Cl)cc2Cn2cncn2)ccc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
CCR2 P41597 1/20 0.39
CCR4 P51679 1/20 0.39
CYP19A1 P11511 5/20 0.38
SLC6A4 P31645 4/20 0.37
HTR2A P28223 3/20 0.37
KCNH2 Q12809 3/20 0.37
SCN9A Q15858 1/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.36
NLRP3 Q96P20 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A3 Q01959 1/20 0.34
STS P08842 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936797 0.90 HTR2A (0.41) CCR1CCR2CCR4CYP19A1SLC6A4
SCHEMBL8936749 0.85 CYP19A1 (0.40) CCR1CCR2CCR4CYP19A1SLC6A4
SCHEMBL8936766 0.84 MAPT (0.41) CCR1CCR2CCR4CYP19A1SLC6A4
SCHEMBL8936805 0.82 CCR1 (0.38) CCR1CCR2CCR4CYP19A1SLC6A4
SCHEMBL8936697 0.78 SLC6A4 (0.39) CYP19A1SLC6A4HTR2AKCNH2SCN9A
SCHEMBL8936735 0.77 PDE7A (0.45) CCR1CCR2CCR4CYP19A1SCN9A
SCHEMBL8936771 0.76 TDP1 (0.41) CCR1CCR2CCR4CYP19A1SLC6A4
SCHEMBL8936779 0.76 SLC6A4 (0.42) CYP19A1SLC6A4HTR2AKCNH2SCN9A
SCHEMBL8936782 0.76 CYP19A1 (0.40) CCR1CCR2CCR4CYP19A1SLC6A4
SCHEMBL8936753 0.74 CYP19A1 (0.41) CCR1CCR2CCR4CYP19A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587392-A THERAPY FOR ESTROGEN DEPENDENT DISEASES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed
EP-0684235-A1 Novel azolyl methyl phenyl derivatives having aromatase inhibitory activity MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1995-11-29 EP disclosed