SCHEMBL8936738

SCHEMBL8936738

COCOc1ccc(C(F)(F)F)cc1CO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
HTT P42858 2/20 0.42
KMT2A Q03164 1/20 0.42
PPARG P37231 3/20 0.42
PPARD Q03181 3/20 0.42
PPARA Q07869 3/20 0.42
PTGDR2 Q9Y5Y4 5/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HPGD P15428 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
FFAR1 O14842 1/20 0.39
FFAR2 O15552 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16959556 0.84 CYP1A2 (0.55) KMT2APPARGPPARDPPARAPTGDR2
SCHEMBL30002156 0.83 HDAC3 (0.49) PPARDPPARAPTGDR2HDAC3HDAC1
SCHEMBL4064597 0.83 HDAC3 (0.49) PPARDPPARAPTGDR2HDAC3HDAC1
SCHEMBL4870587 0.81 KDM4E (0.44) KDM4EHTTKMT2APTGDR2HPGD
SCHEMBL2116117 0.79 MAPK1 (0.41) KDM4EKMT2APTGDR2HPGDALDH1A1
SCHEMBL29953675 0.78 KDM4E (0.42) KDM4EHTTKMT2APTGDR2HDAC3
SCHEMBL16400097 0.77 PTGDR2 (0.66) PPARGPPARDPPARAPTGDR2MAPT
SCHEMBL16961613 0.76 RXRA (0.40) PTGDR2CYP1A2CYP2C9CYP2C19HTR2A
SCHEMBL6211474 0.76 RXRA (0.55) PTGDR2SLC6A4MRGPRX4
SCHEMBL8712221 0.76 PTGDR2 (0.59) KDM4EHTTKMT2APTGDR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587392-A THERAPY FOR ESTROGEN DEPENDENT DISEASES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed
EP-0684235-A1 Novel azolyl methyl phenyl derivatives having aromatase inhibitory activity MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1995-11-29 EP disclosed