SCHEMBL8937642

SCHEMBL8937642

Nc1cc(N)c(-c2ccc([N+](=O)[O-])cc2-c2cccc(Cl)c2Cl)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 3/20 0.44
MAPT P10636 5/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
HPGD P15428 1/20 0.42
S100A4 P26447 2/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
CES1 P23141 1/20 0.41
HSP90AA1 P07900 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
PDE7A Q13946 2/20 0.40
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6049656 0.83 DHFR (0.50) PTPRCMAPTKMT2AMEN1HPGD
SCHEMBL8937640 0.73 PDE7A (0.39) MAPTKMT2AMEN1HPGDPDE7A
SCHEMBL21223480 0.69 NUDT1 (0.45) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL21223471 0.69 FEN1 (0.48) ADRA1A
SCHEMBL435495 0.68 PTPRC (0.85) PTPRCMAPTKMT2AMEN1S100A4
SCHEMBL9755024 0.66 PTPRC (0.62) PTPRCMAPTKMT2AMEN1S100A4
SCHEMBL21223655 0.65 EPHB4 (0.51) HSP90AA1
SCHEMBL7607907 0.65 PDE7A (0.55) PTPRCMAPTKMT2AMEN1S100A4
SCHEMBL10487196 0.65 CYP3A4 (0.64) PTPRCMAPTKMT2AMEN1S100A4
Hydrochloric Acid SCHEMBL21223661 0.64 EPHB4 (0.50) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587380-A ANTIISCHEMIC AGENTS GLAXO WELLCOME INC. (US) 1996-12-24 US disclosed