SCHEMBL8938159

SCHEMBL8938159

O=c1[nH]ncc2cc[c]nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
HSD17B10 Q99714 2/20 0.43
PARP1 P09874 1/20 0.43
PRKCI P41743 1/20 0.43
PDE4B Q07343 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPK1 P28482 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
SLC2A1 P11166 1/20 0.33
HSP90AA1 P07900 1/20 0.31
IDO1 P14902 1/20 0.31
CDK2 P24941 1/20 0.31
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
ADORA2A P29274 1/20 0.31
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
XDH P47989 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL291015 0.74
SCHEMBL15333871 0.72 PARP1 (0.38) PARP1ADORA2A
SCHEMBL19153237 0.72 RAB9A (0.46) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL7366251 0.68 PARP1 (0.53) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL8115281 0.67 ALDH1A1 (0.56) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL18238021 0.64 ALDH1A1 (0.41) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL21388614 0.64 ALDH1A1 (0.41) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL8116183 0.63 HSD17B10 (0.56) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL14911424 0.63 NOS1 (0.56) ALDH1A1HSD17B10PARP1PRKCIPDE4B
SCHEMBL8115175 0.63 ALDH1A1 (0.56) ALDH1A1HSD17B10PARP1PRKCIPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
EP-0612315-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-08-31 EP disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed