SCHEMBL8938826

SCHEMBL8938826

Cc1cc2c(=O)[nH]cc(C)c2cc1OC1CCN(CCC(C)(F)F)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 10/20 0.39
CCR3 P51677 10/20 0.39
ROCK1 Q13464 2/20 0.38
KCNH2 Q12809 3/20 0.36
S1PR5 Q9H228 3/20 0.33
PARP1 P09874 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
ADRA1D P25100 1/20 0.33
CYP2C19 P33261 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
HTR7 P34969 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935557 0.93 HRH1 (0.40) HRH1CCR3ROCK1KCNH2PARP1
SCHEMBL8935395 0.86 PARP1 (0.43) HRH1CCR3ROCK1KCNH2PARP1
SCHEMBL8938757 0.85 ROCK1 (0.56) HRH1CCR3ROCK1KCNH2PARP1
SCHEMBL8935399 0.84 MAOA (0.46) HRH1CCR3ROCK1KCNH2PARP1
SCHEMBL8939164 0.84 ROCK1 (0.57) HRH1CCR3ROCK1KCNH2
SCHEMBL8935441 0.84 HRH1 (0.41) HRH1CCR3ROCK1KCNH2S1PR5
SCHEMBL8935529 0.83 PARP1 (0.44) HRH1CCR3ROCK1KCNH2PARP1
SCHEMBL8934495 0.82 ROCK1 (0.42) HRH1CCR3ROCK1KCNH2PARP1
SCHEMBL8935499 0.82 HRH1 (0.41) HRH1CCR3ROCK1KCNH2S1PR5
SCHEMBL8939077 0.81 HRH1 (0.35) HRH1CCR3KCNH2PARP1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed