SCHEMBL8939077

SCHEMBL8939077

CCc1c[nH]c(=O)c2cc(F)c(OC3CCN(CCC(C)(F)F)CC3)cc12

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 6/20 0.35
CCR3 P51677 6/20 0.35
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
PARP1 P09874 3/20 0.32
DRD2 P14416 1/20 0.31
SLC6A4 P31645 1/20 0.31
NTRK1 P04629 1/20 0.31
TIPARP Q7Z3E1 1/20 0.31
KCNH2 Q12809 1/20 0.31
RET P07949 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937503 0.93 HRH1 (0.35) HRH1CCR3ADRA1DADRA1AADRA1B
SCHEMBL8937316 0.89 DRD2 (0.40) HRH1CCR3PARP1DRD2SLC6A4
SCHEMBL8937313 0.87 MAOA (0.42) HRH1CCR3PARP1DRD2SLC6A4
SCHEMBL8937273 0.87 HRH1 (0.38) HRH1CCR3PARP1KCNH2RET
SCHEMBL8937479 0.85 PARP1 (0.41) HRH1CCR3PARP1DRD2SLC6A4
SCHEMBL8937447 0.84 HRH1 (0.37) HRH1CCR3DRD2SLC6A4KCNH2
SCHEMBL8938999 0.83 PARP1 (0.43) HRH1CCR3PARP1KCNH2MAOA
SCHEMBL8937388 0.83 HRH1 (0.41) HRH1CCR3KCNH2
SCHEMBL8937451 0.83 HRH3 (0.43) HRH1CCR3
SCHEMBL8939065 0.82 HTR1A (0.37) HRH1CCR3ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed