SCHEMBL8941775

SCHEMBL8941775

c1ccc2c(c1)CCc1c-2ccc2c1CCC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
CES1 P23141 1/20 0.47
AKR1B1 P15121 1/20 0.40
BCHE P06276 1/20 0.40
SRD5A1 P18405 1/20 0.40
SRD5A2 P31213 1/20 0.40
PARP1 P09874 1/20 0.40
TSHR P16473 1/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
BCL2L1 Q07817 1/20 0.38
BAD Q92934 1/20 0.38
NOS3 P29474 1/20 0.38
CCNB2 O95067 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNB3 Q8WWL7 1/20 0.38
DRD4 P21917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576506 0.85 PNMT (0.44) CYP2A6MAOAMAOBCES1SRD5A2
SCHEMBL3396448 0.81 TSHR (0.44) CYP2A6MAOAMAOBCES1SRD5A2
SCHEMBL23704623 0.79 PNMT (0.43) CYP2A6MAOAMAOBCES1SRD5A2
SCHEMBL3103992 0.78 CYP2A6 (0.68) CYP2A6MAOAMAOBCES1BCHE
SCHEMBL30505637 0.78 CYP2A6 (0.68) CYP2A6MAOAMAOBCES1BCHE
SCHEMBL17698887 0.77 BCL2L1 (0.54) CYP2A6MAOAMAOBCES1BCHE
SCHEMBL29488244 0.77 BCL2L1 (0.54) CYP2A6MAOAMAOBCES1BCHE
SCHEMBL9652088 0.76 CYP2A6 (0.65) CYP2A6MAOAMAOBCES1BCHE
SCHEMBL30436320 0.76 CYP2A6 (0.65) CYP2A6MAOAMAOBCES1BCHE
SCHEMBL8460056 0.74 CES1 (0.54) CYP2A6MAOAMAOBCES1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480913-A DIHYDRO-PHENANTHRENE DERIVATIVES, SIDE EFFECT REDUCTION ARCH DEVELOPMENT CORPORATION (US) 1996-01-02 US disclosed
EP-0363128-B1 ANTI-ANDROGEN COMPOUNDS ARCH DEVELOPMENT CORPORATION (US) 1993-09-01 EP disclosed
US-5208263-A Dihydrophenanthrene derivatives ARCH DEVELOPMENT CORPORATION (US) 1993-05-04 US disclosed
WO-1990003979-A2 ANTI-ANDROGEN COMPOUNDS ARCH DEVELOPMENT CORPORATION (US) 1990-04-19 WO disclosed
EP-0363128-A2 Anti-androgen compounds ARCH DEVELOPMENT CORPORATION (US) 1990-04-11 EP disclosed