SCHEMBL8942174

SCHEMBL8942174

CC1(N)CN(c2cc3nc4c(cc3cc2F)c(=O)c(C(=O)O)cn4CCF)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LMNA P02545 4/20 0.43
CYP2C9 P11712 1/20 0.43
ATP6V1B2 P21281 1/20 0.43
TBXA2R P21731 1/20 0.43
EDNRA P25101 1/20 0.43
TARBP2 Q15633 1/20 0.43
KDM4E B2RXH2 3/20 0.43
DRD3 P35462 1/20 0.43
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
BRD4 O60885 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
CYP2J2 P51589 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KMT2A Q03164 6/20 0.40
MEN1 O00255 5/20 0.40
NPC1 O15118 1/20 0.40
PIK3CG P48736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942107 0.92 LMNA (0.52) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8941958 0.89 ALDH1A1 (0.39) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942026 0.88 ALDH1A1 (0.44) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL9775969 0.86 ALDH1A1 (0.67) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8941977 0.84 KMT2A (0.38) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8941986 0.84 ALDH1A1 (0.38) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942165 0.84 EPHA2 (0.37) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL9147435 0.84 LMNA (0.58) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8941969 0.84 DPP4 (0.48) ALDH1A1LMNACYP2C9KDM4EHPGD
SCHEMBL8942224 0.83 ALDH1A1 (0.48) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed