SCHEMBL8942224

SCHEMBL8942224

CNC1CN(c2cc3nc4c(cc3cc2F)c(=O)c(C(=O)O)cn4CCF)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.48
TOP1 P11387 3/20 0.46
LMNA P02545 5/20 0.42
CYP2C9 P11712 1/20 0.42
ATP6V1B2 P21281 1/20 0.42
TBXA2R P21731 1/20 0.42
EDNRA P25101 1/20 0.42
TARBP2 Q15633 1/20 0.42
KDM4E B2RXH2 7/20 0.42
DRD3 P35462 1/20 0.42
HPGD P15428 5/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
NPC1 O15118 1/20 0.41
HSD17B10 Q99714 5/20 0.40
HTT P42858 3/20 0.40
TSHR P16473 2/20 0.40
BRD4 O60885 1/20 0.40
CYP2J2 P51589 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942168 0.92 LMNA (0.52) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8942178 0.91 ALDH1A1 (0.47) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8941921 0.90 ALDH1A1 (0.46) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8942358 0.90 ALDH1A1 (0.45) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8941982 0.89 TOP1 (0.43) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8942081 0.89 ALDH1A1 (0.44) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8942041 0.86 TOP1 (0.42) ALDH1A1TOP1LMNACYP2C9ATP6V1B2
SCHEMBL8941960 0.85 DPP4 (0.49) ALDH1A1TOP1LMNACYP2C9KDM4E
SCHEMBL9775969 0.85 ALDH1A1 (0.67) ALDH1A1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942082 0.85 TOP1 (0.41) ALDH1A1TOP1LMNACYP2C9ATP6V1B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed