SCHEMBL8942316

SCHEMBL8942316

O=C(O)c1cn(C2CC2)c2nc3c(F)c(N4CC(N5CCNCC5)C4)c(F)cc3cc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 4/20 0.50
HSD17B10 Q99714 4/20 0.50
HPGD P15428 3/20 0.50
LMNA P02545 3/20 0.50
TOP2A P11388 3/20 0.50
TOP2B Q02880 3/20 0.50
CYP2C9 P11712 2/20 0.50
CYP1A2 P05177 1/20 0.50
DPP4 P27487 6/20 0.47
POLB P06746 2/20 0.44
OPRM1 P35372 2/20 0.44
KCNH2 Q12809 2/20 0.44
PRKD3 O94806 1/20 0.44
ALOX15 P16050 1/20 0.44
CLK2 P49760 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CHRM2 P08172 2/20 0.43
CHRM1 P11229 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9775925 0.92 TOP2A (0.56) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8941990 0.89 LMNA (0.45) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8942324 0.87 LMNA (0.43) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8942130 0.87 LMNA (0.60) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8942137 0.87 LMNA (0.49) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8942301 0.87 LMNA (0.43) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8942162 0.86 DPP4 (0.56) ALDH1A1KDM4EHSD17B10LMNATOP2A
Water SCHEMBL8942213 0.85 DPP4 (0.55) ALDH1A1KDM4EHSD17B10LMNATOP2A
SCHEMBL9775887 0.85 ALDH1A1 (0.62) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL8941979 0.84 DPP4 (0.50) ALDH1A1KDM4EHSD17B10HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed