SCHEMBL8943826

SCHEMBL8943826

CC(C)(C)OC(=O)N(C[C]=O)c1cccc(O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 1/20 0.39
NQO2 P16083 1/20 0.37
F2 P00734 3/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
BRD4 O60885 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
MTNR1A P48039 2/20 0.33
MTNR1B P49286 2/20 0.33
HSD17B1 P14061 2/20 0.33
HSD17B2 P37059 2/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8943566 0.85 ALDH1A1 (0.42) ALDH1A1CYP3A4TSHRF2HDAC1
SCHEMBL4461274 0.85 ALDH1A1 (0.50) ALDH1A1CYP3A4TSHRNQO2F2
SCHEMBL7439248 0.84 MEN1 (0.46) ALDH1A1CYP3A4TSHRF2HDAC1
SCHEMBL8711286 0.83 MIF (0.35) CYP3A4NQO2F2ADRB2ADRB1
SCHEMBL10892391 0.82 ALDH1A1 (0.41) ALDH1A1CYP3A4TSHRNQO2F2
SCHEMBL5648495 0.81 ITGB1 (0.48) ALDH1A1CYP3A4TSHRNQO2F2
SCHEMBL7437218 0.80 MEN1 (0.38) ALDH1A1NQO2F2MTNR1AMTNR1B
SCHEMBL8707172 0.78 MT-CO2 (0.35) ALDH1A1TSHRHDAC1HDAC6ITGB1
SCHEMBL9222980 0.76 KCNQ4 (0.41) HDAC1HDAC8HDAC6ADRB2ADRB1
SCHEMBL8712805 0.75 KDM4E (0.40) ALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532353-A Process for the preparation of halogenated β-lactam compounds BIOCHIMICA OPOS SPA (IT) 1996-07-02 US disclosed
EP-0570058-A2 Process for the preparation of halogenated beta-lactam compounds BIOCHIMICA OPOS SPA (IT) 1993-11-18 EP disclosed