SCHEMBL8944351

SCHEMBL8944351

O=C1CCc2c(ccc3ccccc23)N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.47
CYP2C9 P11712 2/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP1A2 P05177 2/20 0.47
HPGD P15428 2/20 0.47
GLA P06280 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NPC1 O15118 1/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
MAPK14 Q16539 1/20 0.47
TP53 P04637 3/20 0.46
CYP2D6 P10635 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
CYP2B6 P20813 1/20 0.45
MAPT P10636 3/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050070 0.90 MAPT (0.50) CYP2C19CYP2C9KDM4ECYP1A2HPGD
Sulfuric Acid SCHEMBL8944460 0.89 PKM (0.43) CYP2C19CYP2C9KDM4ECYP1A2HPGD
SCHEMBL29124061 0.84 CDK5 (0.47) CYP2C19KDM4ECYP1A2HPGDSIRT1
SCHEMBL8944299 0.77 AHR (0.46) MAPTCDK5CDK5R1PKMKIF11
SCHEMBL8714752 0.76 KDM4E (0.41) CYP2C19CYP2C9KDM4ECYP1A2HPGD
SCHEMBL1287805 0.75 CYP11B1 (0.47) CYP2C19CYP2C9KDM4ECYP1A2HPGD
SCHEMBL15801195 0.75 PNMT (0.45) CYP2C9KDM4ECYP1A2HPGDHSD17B10
SCHEMBL8715073 0.74 TP53 (0.40) CYP2C19CYP2C9KDM4ECYP1A2HPGD
SCHEMBL8713911 0.74 ANPEP (0.44) CYP2C19CYP2C9KDM4ECYP1A2HPGD
Hydrochloric Acid SCHEMBL8717493 0.73 ANPEP (0.43) CYP2C19CYP2C9KDM4ECYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489215-A1 PROCESS FOR PRODUCING ORGANIC COMPOUND Kaneka Corporation (JP) 2019-05-29 EP disclosed
EP-0724440-A4 DI- AND TETRA-HYDROBENZO F]QUINOLIN-3-ONES SMITHKLINE BEECHAM CORP (US) 1996-11-20 EP disclosed
EP-0724440-A1 DI- AND TETRA-HYDROBENZO F]QUINOLIN-3-ONES SMITHKLINE BEECHAM CORPORATION (US) 1996-08-07 EP disclosed
WO-1995005821-A1 DI- AND TETRA-HYDROBENZO[F]QUINOLIN-3-ONES SMITHKLINE BEECHAM CORPORATION (US) 1995-03-02 WO disclosed