SCHEMBL8944521

SCHEMBL8944521

O=C(O)c1ccccc1-c1ccc(Cn2c(-c3ccccn3)nc3ccccc32)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.63
AGTR1 P30556 2/20 0.61
AGTR2 P50052 2/20 0.61
CTSD P07339 4/20 0.58
L3MBTL1 Q9Y468 1/20 0.57
GRM2 Q14416 1/20 0.57
KDM4E B2RXH2 3/20 0.53
CYP2C9 P11712 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
GUSB P08236 2/20 0.53
HRH3 Q9Y5N1 1/20 0.52
ALDH1A1 P00352 2/20 0.52
HSD17B10 Q99714 2/20 0.52
ABCC3 O15438 1/20 0.52
ABCC4 O15439 1/20 0.52
USP2 O75604 1/20 0.52
ABCB11 O95342 1/20 0.52
CHRM2 P08172 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8391622 0.88 PPARG (0.69) PPARGAGTR1AGTR2L3MBTL1KDM4E
SCHEMBL9041351 0.86 GRM2 (0.56) PPARGAGTR1AGTR2CTSDL3MBTL1
SCHEMBL8394581 0.85 GRM2 (0.52) PPARGAGTR1AGTR2CTSDL3MBTL1
SCHEMBL8392673 0.85 PPARG (0.66) PPARGAGTR1AGTR2KDM4ECYP2C9
SCHEMBL8944506 0.85 KDM4E (0.62) PPARGAGTR1AGTR2KDM4ECYP2C9
SCHEMBL8393577 0.83 PPARG (0.61) PPARGAGTR1AGTR2GRM2KDM4E
SCHEMBL8396864 0.83 PPARG (0.72) PPARGAGTR1AGTR2
SCHEMBL230485 0.83 ALDH1A1 (0.66) CTSDL3MBTL1KDM4ECYP2C9CYP1A2
SCHEMBL29411979 0.83 ALDH1A1 (0.66) CTSDL3MBTL1KDM4ECYP2C9CYP1A2
SCHEMBL8391717 0.82 PPARG (0.71) PPARGAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541229-A ANGIOITENSIN II ANTAGONIST AS HYPOTENSIVE AGENTS, ANTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0392317-B1 Benzimidazoles, drugs containing these compounds and process for their preparation THOMAE GMBH DR K (DE) 1996-01-03 EP disclosed