SCHEMBL8944545

SCHEMBL8944545

CN1CCN(Cc2ccc(Cl)cc2Cl)C(C2(C)NCCN2)C1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
CYP2A13 Q16696 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
P2RX7 Q99572 6/20 0.35
TSHR P16473 1/20 0.35
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036088 0.74 KDM4E (0.45) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL2387265 0.72 KDM4E (0.44) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL8944590 0.70 KDM4E (0.45) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL9036092 0.69 KDM4E (0.45) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL8944705 0.69 TSHR (0.56) KDM4ETDP1ALDH1A1POLBP2RX7
SCHEMBL8944840 0.69 KDM4E (0.43) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL2656580 0.68 KDM4E (0.88) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL29604869 0.66 KDM4E (0.42) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL28368198 0.65 CYP2A13 (0.43) KDM4ETDP1ALDH1A1POLBCYP2A13
SCHEMBL593572 0.62 CYP2A13 (0.66) KDM4ETDP1ALDH1A1POLBCYP2A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500426-A ADMINISTERED TO IMPROVE GLUCOSE TOLERANCE ADIR ET COMPAGNIE (FR) 1996-03-19 US disclosed
US-5492912-A IMPROVES GLUCOSE TOLERANCE ADIR ET COMPAGNIE (FR) 1996-02-20 US disclosed
EP-0638568-A1 Substituted piperazines, their process of preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1995-02-15 EP disclosed