SCHEMBL8944906

SCHEMBL8944906

NC(=O)OCC(N)COc1noc2ccc(Br)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 3/20 0.34
TP53 P04637 2/20 0.34
HSD17B10 Q99714 2/20 0.34
FAAH O00519 1/20 0.34
TSHR P16473 3/20 0.33
MAPT P10636 2/20 0.33
CA12 O43570 2/20 0.32
CA9 Q16790 2/20 0.32
PIM1 P11309 1/20 0.32
ALDH1A1 P00352 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
SIRT1 Q96EB6 1/20 0.31
KMT2A Q03164 2/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945107 0.86 FAAH (0.49) CYP1A2KDM4ETP53HSD17B10FAAH
Hydrochloric Acid SCHEMBL8945306 0.86 FAAH (0.34) CYP1A2KDM4EFAAHMAPTSMN1; SMN2
SCHEMBL8945254 0.86 FAAH (0.34) CYP1A2KDM4EFAAHSMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL8945060 0.85 FAAH (0.48) CYP1A2KDM4ETP53HSD17B10FAAH
SCHEMBL8945175 0.83 TBK1 (0.33) CYP1A2KDM4EFAAHSMN1; SMN2LMNA
SCHEMBL8945191 0.83 KCNH2 (0.40) CYP1A2KDM4EHSD17B10MAPTALDH1A1
SCHEMBL8944960 0.83 FAAH (0.45) CYP1A2KDM4ETP53HSD17B10FAAH
Hydrochloric Acid SCHEMBL8945351 0.82 FAAH (0.34) CYP1A2KDM4EFAAHMAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL8945170 0.82 FAAH (0.38) CYP1A2KDM4ETP53FAAHTSHR
Hydrochloric Acid SCHEMBL8945261 0.82 FAAH (0.44) CYP1A2KDM4ETP53HSD17B10FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578627-A FOR TREATING CEREBRAL CIRCULATORY DISORDER, HEAD INJURY SEQUELAE AND/OR EPILEPSY TOYAMA CHEMICAL CO., LTD. (JP) 1996-11-26 US disclosed
EP-0665226-A1 NOVEL 1,2-BENZISOXAZOLE DERIVATIVE OR SALT THEREOF, AND BRAIN PROTECTIVE AGENT COMPRISING THE SAME TOYAMA CHEMICAL CO., LTD. (JP) 1995-08-02 EP disclosed