SCHEMBL8945191

SCHEMBL8945191

NC(=O)OCC(N)COc1noc2ccc(-c3ccccc3)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.40
SCN5A Q14524 1/20 0.39
NPC1 O15118 2/20 0.38
KDM4E B2RXH2 3/20 0.37
CYP1A2 P05177 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP2D6 P10635 1/20 0.36
PKM P14618 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
HIF1A Q16665 1/20 0.35
SLC1A5 Q15758 1/20 0.35
LMNA P02545 1/20 0.34
IP6K1 Q92551 1/20 0.34
ACACA Q13085 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8944960 0.85 FAAH (0.45) NPC1KDM4ECYP1A2SMN1; SMN2CYP2D6
Hydrochloric Acid SCHEMBL8945261 0.84 FAAH (0.44) NPC1KDM4ECYP1A2SMN1; SMN2CYP2D6
Hydrochloric Acid SCHEMBL8945510 0.84 FAAH (0.44) NPC1KDM4ECYP1A2SMN1; SMN2CYP2D6
SCHEMBL8945107 0.83 FAAH (0.49) KCNH2SCN5AKDM4ECYP1A2SMN1; SMN2
SCHEMBL8944906 0.83 CYP1A2 (0.35) KDM4ECYP1A2SMN1; SMN2CYP2D6PKM
SCHEMBL8945254 0.83 FAAH (0.34) KCNH2KDM4ECYP1A2SMN1; SMN2CYP2D6
Hydrochloric Acid SCHEMBL8945306 0.83 FAAH (0.34) KCNH2NPC1KDM4ECYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL8945060 0.82 FAAH (0.48) KCNH2SCN5AKDM4ECYP1A2SMN1; SMN2
SCHEMBL8945175 0.80 TBK1 (0.33) KDM4ECYP1A2SMN1; SMN2LMNATBK1
Hydrochloric Acid SCHEMBL8945170 0.80 FAAH (0.38) KDM4ECYP1A2SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578627-A FOR TREATING CEREBRAL CIRCULATORY DISORDER, HEAD INJURY SEQUELAE AND/OR EPILEPSY TOYAMA CHEMICAL CO., LTD. (JP) 1996-11-26 US disclosed
EP-0665226-A1 NOVEL 1,2-BENZISOXAZOLE DERIVATIVE OR SALT THEREOF, AND BRAIN PROTECTIVE AGENT COMPRISING THE SAME TOYAMA CHEMICAL CO., LTD. (JP) 1995-08-02 EP disclosed