SCHEMBL8945121

SCHEMBL8945121

CC(C)(C)OC(=O)Nc1ccc2onc(OCC(COC(N)=O)NC(=O)OC(C)(C)C)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
MAP4K4 O95819 1/20 0.38
AURKA O14965 2/20 0.36
RPS6KB1 P23443 2/20 0.36
AAK1 Q2M2I8 6/20 0.36
JAK2 O60674 2/20 0.35
HDAC1 Q13547 4/20 0.35
HDAC3 O15379 3/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC6 Q9UBN7 3/20 0.35
HDAC10 Q969S8 2/20 0.35
EGFR P00533 3/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945202 0.89 CA12 (0.41) CA12CA1CA9MAP4K4AURKA
SCHEMBL8945081 0.88 FAAH (0.43) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945043 0.86 CTSS (0.37) CA1CA9AAK1HDAC1HDAC3
SCHEMBL8945143 0.84 AAK1 (0.35) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8944963 0.80 FAAH (0.41) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8944929 0.80 FAAH (0.42) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945028 0.80 FAAH (0.42) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945072 0.79 FAAH (0.43) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945356 0.79 AAK1 (0.38) AAK1JAK2HDAC1HDAC3HDAC2
SCHEMBL8945585 0.78 AAK1 (0.40) MAP4K4AAK1JAK2HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578627-A FOR TREATING CEREBRAL CIRCULATORY DISORDER, HEAD INJURY SEQUELAE AND/OR EPILEPSY TOYAMA CHEMICAL CO., LTD. (JP) 1996-11-26 US disclosed
EP-0665226-A1 NOVEL 1,2-BENZISOXAZOLE DERIVATIVE OR SALT THEREOF, AND BRAIN PROTECTIVE AGENT COMPRISING THE SAME TOYAMA CHEMICAL CO., LTD. (JP) 1995-08-02 EP disclosed