SCHEMBL8945202

SCHEMBL8945202

CC(C)(C)OC(=O)Nc1ccc2onc(OCC(CO)NC(=O)OC(C)(C)C)c2c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA9 Q16790 1/20 0.41
AAK1 Q2M2I8 6/20 0.40
MAP4K4 O95819 1/20 0.38
HDAC1 Q13547 5/20 0.37
HDAC3 O15379 3/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 4/20 0.36
HDAC10 Q969S8 2/20 0.36
EGFR P00533 4/20 0.36
JAK2 O60674 1/20 0.35
CYP17A1 P05093 1/20 0.35
AURKA O14965 1/20 0.35
RPS6KB1 P23443 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945356 0.90 AAK1 (0.38) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945121 0.89 CA12 (0.38) CA12CA1CA9AAK1MAP4K4
SCHEMBL8944950 0.87 FAAH (0.46) AAK1
SCHEMBL8945585 0.87 AAK1 (0.40) AAK1MAP4K4HDAC1HDAC3HDAC2
SCHEMBL8945110 0.85 CTSS (0.39) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945382 0.85 SSTR4 (0.44) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945097 0.83 AAK1 (0.38) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945482 0.80 FAAH (0.44) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8945072 0.76 FAAH (0.43) AAK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8944941 0.76 FAAH (0.43) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578627-A FOR TREATING CEREBRAL CIRCULATORY DISORDER, HEAD INJURY SEQUELAE AND/OR EPILEPSY TOYAMA CHEMICAL CO., LTD. (JP) 1996-11-26 US disclosed
EP-0665226-A1 NOVEL 1,2-BENZISOXAZOLE DERIVATIVE OR SALT THEREOF, AND BRAIN PROTECTIVE AGENT COMPRISING THE SAME TOYAMA CHEMICAL CO., LTD. (JP) 1995-08-02 EP disclosed