SCHEMBL8945875

SCHEMBL8945875

CNC(Cc1cc(Br)cc(Br)c1N)c1sccc1C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.32
SLC6A4 P31645 2/20 0.32
KCNH2 Q12809 2/20 0.32
LMNA P02545 2/20 0.32
GBA1 P04062 1/20 0.32
CYP1A2 P05177 1/20 0.32
CNR1 P21554 1/20 0.32
TBXA2R P21731 1/20 0.32
HRH2 P25021 1/20 0.32
HIF1A Q16665 1/20 0.32
ABCB11 O95342 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
AR P10275 1/20 0.32
SLC6A2 P23975 1/20 0.32
PDE4A P27815 1/20 0.32
SLC6A3 Q01959 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
CYP3A4 P08684 2/20 0.32
HTT P42858 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8946047 0.99 CYP3A4 (0.33) CYP2D6SLC6A4KCNH2LMNAGBA1
SCHEMBL9425401 0.84 MAPT (0.30)
SCHEMBL8945857 0.81 ALDH1A1 (0.32) CYP1A2HIF1AALOX15
SCHEMBL8946076 0.75 TDP1 (0.35) SLC6A4CYP3A4ALOX15TDP1
SCHEMBL8945809 0.75 TDP1 (0.33) CYP3A4ALOX15TDP1
SCHEMBL8946017 0.75 ALOX5 (0.33) CYP3A4TDP1
SCHEMBL8946111 0.74 CYP3A4 (0.39) SLC6A4KCNH2CYP3A4HTTALOX15
SCHEMBL8946168 0.73 SLC6A2 (0.40) SLC6A4SLC6A2
SCHEMBL8946019 0.73 MEN1 (0.32)
SCHEMBL8945970 0.73 CYP3A4 (0.35) CYP3A4HTTALOX15TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed