SCHEMBL8945857

SCHEMBL8945857

CNC(Cc1ccc(Br)cc1N)c1sccc1C

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
ALOX15 P16050 1/20 0.32
CASP7 P55210 1/20 0.32
HIF1A Q16665 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALOX5 P09917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9425401 0.90 MAPT (0.30) ALOX5
SCHEMBL8946076 0.87 TDP1 (0.35) ALDH1A1ALOX15ALOX5
SCHEMBL8946111 0.86 CYP3A4 (0.39) ALDH1A1ALOX15ALOX5
SCHEMBL8946080 0.85 MEN1 (0.32) ALOX5
Hydrochloric Acid SCHEMBL8946071 0.85 CYP3A4 (0.38) ALDH1A1ALOX15
SCHEMBL8946168 0.85 SLC6A2 (0.40) ALOX5
SCHEMBL8946175 0.82 MEN1 (0.34) ALDH1A1
SCHEMBL8946001 0.81 ALDH1A1 (0.34) ALDH1A1HSD17B10
SCHEMBL8946017 0.81 ALOX5 (0.33) ALDH1A1ALOX5
SCHEMBL8945875 0.81 CYP2D6 (0.32) CYP1A2ALOX15HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed