SCHEMBL8945886

SCHEMBL8945886

CNC(Cc1cc(C(F)(F)F)ccc1N)c1sccc1C

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
GFER P55789 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CFTR P13569 1/20 0.31
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8946060 0.99 HTR2A (0.32) HTR2ASLC6A4KCNH2KDM4EMEN1
SCHEMBL8946001 0.91 ALDH1A1 (0.34) SLC6A4KDM4EMEN1ALDH1A1GAA
SCHEMBL8946019 0.84 MEN1 (0.32) MEN1ALDH1A1GAAKMT2AL3MBTL1
SCHEMBL8945809 0.84 TDP1 (0.33) ALDH1A1
SCHEMBL8946130 0.81 SLC6A2 (0.32) SLC6A4
SCHEMBL9425401 0.81 MAPT (0.30) MAPT
SCHEMBL8945970 0.81 CYP3A4 (0.35) ALDH1A1
SCHEMBL8946128 0.80 HTR2A (0.35) HTR2AALDH1A1
SCHEMBL9425059 0.79 NPC1 (0.35) ALDH1A1MAPTL3MBTL1
SCHEMBL8946017 0.78 ALOX5 (0.33) KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed