SCHEMBL8945924

SCHEMBL8945924

CCCCCC(N)Cc1ccccc1N

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CSNK1E P49674 1/20 0.43
SIGMAR1 Q99720 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR2A P28223 1/20 0.37
PLA2G1B P04054 1/20 0.37
PLA2G2A P14555 1/20 0.37
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4557993 0.83 CSNK1E (0.43) CSNK1ECYP1A2CYP2C9CYP2C19
SCHEMBL28036434 0.80 CSNK1E (0.48) CSNK1ESIGMAR1
SCHEMBL21800790 0.80 CSNK1E (0.48) CSNK1ESIGMAR1
SCHEMBL11120190 0.80 CSNK1E (0.48) CSNK1ESIGMAR1
SCHEMBL7513002 0.80 HTR2A (0.50) HTR2A
SCHEMBL24148832 0.79 SIGMAR1 (0.40) CSNK1ESIGMAR1HTR2A
SCHEMBL15579942 0.77 CSNK1E (0.68) CSNK1ESIGMAR1
SCHEMBL3840317 0.77 CSNK1E (0.68) CSNK1ESIGMAR1
SCHEMBL543510 0.76 ALDH1A1 (0.42) CYP1A2CYP2C9CYP2C19
SCHEMBL29289210 0.75 HTR2A (0.41) CSNK1ESIGMAR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed