SCHEMBL8945925

SCHEMBL8945925

CC(C)C1=Nc2ccccc2CC(c2ccsc2)N1C

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRK1 P41145 1/20 0.31
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945951 0.98 ADORA2B (0.31) ADORA2B
SCHEMBL8945994 0.84 HSD17B10 (0.34) ADORA2BHRH4
SCHEMBL8946148 0.81 ADORA2B (0.33) ADORA2BOPRM1OPRK1HRH4
SCHEMBL8945923 0.81 HRH4 (0.35) HRH4
Hydrochloric Acid SCHEMBL8945921 0.80 HRH4 (0.34) HRH4
Hydrochloric Acid SCHEMBL8945865 0.80 ADORA2B (0.32) ADORA2BOPRM1OPRK1
SCHEMBL8946091 0.79 SLC6A2 (0.38) HRH4
SCHEMBL8945861 0.79 SMN1; SMN2 (0.32) ADORA2B
Hydrochloric Acid SCHEMBL8945737 0.78 SLC6A2 (0.37) HRH4
SCHEMBL8946123 0.78 OPRM1 (0.31) ADORA2BOPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed