SCHEMBL8946115

SCHEMBL8946115

CNC(Cc1ccccc1N)c1cc(C)cs1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
CXCR1 P25024 1/20 0.30
CXCR2 P25025 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945903 0.78 LTA4H (0.36) SLC6A2SLC6A4SLC6A3
SCHEMBL8945765 0.77 CYP3A4 (0.33) SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL8945808 0.76 LTA4H (0.37) SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL8945802 0.76 LTA4H (0.37) SLC6A2SLC6A4SLC6A3
SCHEMBL8946102 0.75 SLC6A2 (0.37) SLC6A2SLC6A4
SCHEMBL10565227 0.75 GAA (0.38) SLC6A4
SCHEMBL8945959 0.74 HDAC1 (0.35) SLC6A3
SCHEMBL8945855 0.74 HDAC1 (0.35) SLC6A3
Hydrochloric Acid SCHEMBL9582349 0.74 TDP1 (0.37)
SCHEMBL8945781 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed