SCHEMBL8945855

SCHEMBL8945855

CNC(Cc1ccccc1N)c1cnc(C)s1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
SLC6A3 Q01959 1/20 0.32
GUCY1B2 O75343 1/20 0.31
GUCY1A2 P33402 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945765 0.79 CYP3A4 (0.33) SLC6A3
SCHEMBL8945917 0.78 NOS1 (0.34) HDAC1SLC6A3
SCHEMBL8946102 0.77 SLC6A2 (0.37)
SCHEMBL8945905 0.75 YTHDC1 (0.33)
SCHEMBL8945903 0.74 LTA4H (0.36) SLC6A3
SCHEMBL8946115 0.74 SLC6A2 (0.31) SLC6A3
SCHEMBL8945959 0.73 HDAC1 (0.35) HDAC1HDAC2SLC6A3
Hydrochloric Acid SCHEMBL8945808 0.72 LTA4H (0.37) SLC6A3
Hydrochloric Acid SCHEMBL8945802 0.72 LTA4H (0.37) SLC6A3
SCHEMBL8945955 0.71 TSHR (0.38) SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed