SCHEMBL8945903

SCHEMBL8945903

CNC(Cc1ccccc1N)c1cccs1

nearest known ligand 0.97

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.36
SLC6A2 P23975 4/20 0.33
SLC6A4 P31645 4/20 0.33
SLC6A3 Q01959 4/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
KCNH2 Q12809 3/20 0.33
MLNR O43193 1/20 0.33
CACNA1F O60840 1/20 0.33
CYP1A2 P05177 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR1A P08908 1/20 0.33
GAA P10253 1/20 0.33
CYP2C9 P11712 1/20 0.33
DRD2 P14416 1/20 0.33
KCNE1 P15382 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945808 0.97 LTA4H (0.37) LTA4HSLC6A2SLC6A4SLC6A3CYP3A4
Hydrochloric Acid SCHEMBL8945802 0.97 LTA4H (0.37) LTA4HSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL8946102 0.78 SLC6A2 (0.37) SLC6A2SLC6A4HRH1
SCHEMBL8946115 0.78 SLC6A2 (0.31) SLC6A2SLC6A4SLC6A3
SCHEMBL8945765 0.78 CYP3A4 (0.33) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8946017 0.77 ALOX5 (0.33) CYP3A4KMT2A
SCHEMBL8945781 0.77
Hydrochloric Acid SCHEMBL9482649 0.76 TAAR1 (0.46) CYP3A4CYP2D6CYP2C19
SCHEMBL9001661 0.76 ALDH1A1 (0.42) HTR2AADRA1AHRH1
Hydrochloric Acid SCHEMBL8945916 0.75 CYP3A4 (0.30) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed