SCHEMBL8946775

SCHEMBL8946775

CC1(C)Oc2ccc(I)cc2[C@@H](N)[C@@H]1O

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 8/20 0.37
KCNQ1 P51787 8/20 0.37
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
ABCB1 P08183 7/20 0.35
ABCC9 O60706 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
KCND3 Q9UK17 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946767 1.00 KCNE1 (0.37) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL8946770 1.00 KCNE1 (0.37) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9197856 0.82 HTR1A (0.39) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9197846 0.82 HTR1A (0.39) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9197844 0.82 HTR1A (0.39) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9198451 0.81 KCNE1 (0.37) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9032549 0.81 KCNE1 (0.56) KCNE1KCNQ1ABCC9
SCHEMBL9530286 0.81 KCNE1 (0.53) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9530280 0.81 KCNE1 (0.53) KCNE1KCNQ1KDM4EL3MBTL1ABCB1
SCHEMBL9198446 0.81 KCNE1 (0.37) KCNE1KCNQ1KDM4EL3MBTL1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500442-A Cyclobut-3-ene-1,2-dione derivatives as smooth muscle relaxants AMERICAN HOME PRODUCTS CORPORATION (US) 1996-03-19 US disclosed