SCHEMBL8946969

SCHEMBL8946969

NC1C(=O)N(CC(=O)N2CCCC2)c2ccccc2N(C2CCCCC2)C1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 4/20 0.61
CCKBR P32239 4/20 0.61
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GFER P55789 1/20 0.44
RAB9A P51151 1/20 0.43
POLB P06746 1/20 0.43
CHRM2 P08172 3/20 0.43
CHRM4 P08173 3/20 0.43
CHRM1 P11229 3/20 0.43
CHRM3 P20309 2/20 0.43
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468864 0.88 ALDH1A1 (0.58) CCKARCCKBRALDH1A1MEN1KMT2A
SCHEMBL6180507 0.81 CCKAR (0.51) CCKARCCKBRALDH1A1MEN1KMT2A
SCHEMBL8946837 0.77 CCKBR (0.62) CCKARCCKBRALDH1A1MEN1KMT2A
SCHEMBL14520869 0.77 CCKBR (1.00) CCKARCCKBR
SCHEMBL8946676 0.77 CCKBR (1.00) CCKARCCKBR
SCHEMBL8946830 0.75 CCKBR (0.74) CCKARCCKBR
SCHEMBL7088452 0.73 CHRM2 (0.58) CCKBRALDH1A1MEN1KMT2ACHRM2
SCHEMBL8865990 0.73 CCKBR (0.63) CCKBR
SCHEMBL4075043 0.72 CHRM2 (0.56) CCKBRALDH1A1MEN1KMT2APOLB
SCHEMBL8691247 0.72 HTT (0.38) CCKARALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585376-A 1,5-benzodiazepine derivatives having CCK and/or gastrin antagonistic activity GLAXO WELLCOME INC. (US) 1996-12-17 US disclosed