SCHEMBL8947322

SCHEMBL8947322

CS(=O)(=O)c1ccc(-c2nnnn2CC(=O)O)cc1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.66
HPGD P15428 1/20 0.66
PTGS2 P35354 10/20 0.52
HSP90AA1 P07900 1/20 0.48
LMNA P02545 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.43
TP53 P04637 1/20 0.43
HSD11B1 P28845 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947331 0.87 ALDH1A1 (0.84) ALDH1A1HPGDLMNAHSD11B1
SCHEMBL8947309 0.85 HSP90AA1 (0.53) ALDH1A1HPGDPTGS2HSP90AA1LMNA
SCHEMBL5966727 0.84 ALDH1A1 (0.75) ALDH1A1HPGDPTGS2HSD11B1
SCHEMBL8947338 0.83 ALDH1A1 (0.59) ALDH1A1HPGDPTGS2HSP90AA1HSD11B1
SCHEMBL8947261 0.81 ALDH1A1 (0.75) ALDH1A1HPGDHSD11B1
SCHEMBL8947281 0.81 ALDH1A1 (0.75) ALDH1A1HPGDHSD11B1
SCHEMBL5966693 0.81 ALDH1A1 (0.74) ALDH1A1HPGDHSD11B1
SCHEMBL8947199 0.80 ALDH1A1 (0.73) ALDH1A1HPGDHSD11B1
SCHEMBL8947164 0.80 ALDH1A1 (1.00) ALDH1A1HPGDPTGS2HSD11B1
SCHEMBL8947260 0.80 ALDH1A1 (0.73) ALDH1A1HPGDPTGS2LMNAHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35281-E ANTIDIABETIC AGENTS WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
EP-0388967-B1 Aldose reductase inhibitor WAKAMOTO PHARMA CO LTD (JP) 1995-06-28 EP disclosed
US-5055481-A Alleviate diabetic complications WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1991-10-08 US disclosed
EP-0388967-A1 Aldose reductase inhibitor Wakamoto Pharmaceutical Co., Ltd. (JP) 1990-09-26 EP disclosed