SCHEMBL8947309

SCHEMBL8947309

COC(=O)Cn1nnnc1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.53
PTGS2 P35354 10/20 0.51
HSP90B1 P14625 1/20 0.51
TRAP1 Q12931 1/20 0.51
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.48
TRPV1 Q8NER1 1/20 0.46
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947317 0.89 ALDH1A1 (0.57) ALDH1A1HPGDTRPV1LMNA
SCHEMBL8947251 0.85 TRPV1 (0.45) HSP90AA1PTGS2HSP90B1TRAP1ALDH1A1
SCHEMBL8947322 0.85 ALDH1A1 (0.66) HSP90AA1PTGS2ALDH1A1HPGDLMNA
SCHEMBL8947240 0.85 ALDH1A1 (0.54) ALDH1A1HPGDTRPV1
SCHEMBL8947310 0.83 TRPV1 (0.63) ALDH1A1HPGDTRPV1LMNA
SCHEMBL8947140 0.83 HSD11B1 (0.59) PTGS2ALDH1A1HPGDTRPV1LMNA
SCHEMBL8947278 0.83 ALDH1A1 (0.70) PTGS2ALDH1A1HPGDTRPV1
SCHEMBL8947311 0.83 ALDH1A1 (0.57) PTGS2ALDH1A1HPGDTRPV1
SCHEMBL8947149 0.83 ALDH1A1 (0.51) ALDH1A1HPGDTRPV1LMNA
SCHEMBL5966689 0.82 TRPV1 (0.59) ALDH1A1HPGDTRPV1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35281-E ANTIDIABETIC AGENTS WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
EP-0388967-B1 Aldose reductase inhibitor WAKAMOTO PHARMA CO LTD (JP) 1995-06-28 EP disclosed
US-5055481-A Alleviate diabetic complications WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1991-10-08 US disclosed
EP-0388967-A1 Aldose reductase inhibitor Wakamoto Pharmaceutical Co., Ltd. (JP) 1990-09-26 EP disclosed