SCHEMBL8947994

SCHEMBL8947994

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)sc3cc(CCCCN4CCN(c5cccc6ccccc56)CC4)ccc32)CC1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
HTR2A P28223 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CYP2D6 P10635 1/20 0.51
HTR1A P08908 3/20 0.50
HTR2C P28335 3/20 0.50
SIGMAR1 Q99720 2/20 0.47
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
DRD2 P14416 1/20 0.45
HPGD P15428 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
DRD1 P21728 1/20 0.45
DRD4 P21917 1/20 0.45
HTR1D P28221 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948074 0.90 HTR1A (0.53) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8947933 0.89 HTR1A (0.66) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8948013 0.89 HTR1A (0.56) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8947985 0.88 KDM4E (0.58) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8947779 0.86 KDM4E (0.54) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8947998 0.84 HTR2A (0.46) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8948078 0.84 HTR2A (0.55) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8947762 0.84 HTR1A (0.66) CYP1A2CYP3A4HTR2AKDM4ECYP2D6
SCHEMBL8948192 0.83 HTR1A (0.65) HTR2AHTR1AHTR2CHTR7
SCHEMBL7765360 0.83 HTR2A (0.47) CYP1A2CYP3A4HTR2AKDM4ECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed