SCHEMBL8947998

SCHEMBL8947998

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)sc3cc(CCCCN4CCNCC4c4cccc5ccccc45)ccc32)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.46
CYP1A2 P05177 3/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HTR2C P28335 3/20 0.44
HTR1A P08908 2/20 0.44
CYP2C9 P11712 2/20 0.44
DRD2 P14416 2/20 0.44
HPGD P15428 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
HTR7 P34969 2/20 0.44
HTR6 P50406 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947994 0.84 CYP1A2 (0.51) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8948078 0.80 HTR2A (0.55) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8947985 0.80 KDM4E (0.58) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8947898 0.79 HTR2A (0.55) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8947779 0.77 KDM4E (0.54) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8948074 0.77 HTR1A (0.53) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8947974 0.77 SIGMAR1 (0.64) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8948030 0.77 SIGMAR1 (0.62) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8948013 0.76 HTR1A (0.56) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL8947933 0.76 HTR1A (0.66) HTR2ACYP1A2CYP3A4CYP2D6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed