SCHEMBL8948073

SCHEMBL8948073

CCCN(CCC)CCc1cc2sc(=O)[nH]c2cc1OC

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
MKNK1 Q9BUB5 4/20 0.38
HTR1A P08908 3/20 0.38
HTR2C P28335 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947871 0.75 DRD2 (0.48) PDE3BPDE3AHTR1AHTR2C
SCHEMBL11206860 0.74 PDE3B (0.61) PDE3BPDE3AMKNK1HTR1AHTR2C
SCHEMBL11336169 0.70 PDE3B (0.56) PDE3BPDE3AMKNK1HTR1AHTR2C
SCHEMBL7762986 0.70 HTR1A (0.45) PDE3BPDE3AHTR1AHTR2C
SCHEMBL15534441 0.69 PDE3B (0.54) PDE3BPDE3AMKNK1HTR1AHTR2C
SCHEMBL8948133 0.69 HTR1A (0.53) HTR1AHTR2C
SCHEMBL10986865 0.69 DRD2 (0.47) HTR1A
Hydrochloric Acid SCHEMBL10867793 0.68 APEX1 (0.48) HTR1A
Hydrochloric Acid SCHEMBL10754007 0.67 HTR1A (0.38) HTR1AHTR2C
SCHEMBL11347101 0.66 PDE3B (0.54) PDE3BPDE3AMKNK1HTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed