SCHEMBL8948104

SCHEMBL8948104

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)oc3cc(CCCCN4CCN(c5cccc(C(F)(F)F)c5)CC4)ccc32)CC1

nearest known ligand 0.76

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52
HTR1A P08908 3/20 0.52
KDM4E B2RXH2 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
SIGMAR1 Q99720 1/20 0.47
HTR2C P28335 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947762 0.86 HTR1A (0.66) HTR2AHTR1AKDM4ECYP1A2CYP3A4
SCHEMBL8947873 0.84 HTR2A (0.56) HTR2ASLC6A2SLC6A4SLC6A3KDM4E
SCHEMBL8947957 0.83 HTR1A (0.65) HTR2ASLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8948076 0.81 HTR1A (0.64) HTR2AHTR1ACYP1A2CYP3A4CYP2D6
SCHEMBL8948109 0.79 HTR2A (0.61) HTR2AHTR1AKDM4ECYP1A2CYP3A4
SCHEMBL7766399 0.78 HTR2A (0.49) HTR2ASLC6A2SLC6A4SLC6A3HTR2C
SCHEMBL10394830 0.76 HTR1A (0.65) HTR2ASLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8947985 0.76 KDM4E (0.58) HTR2AHTR1AKDM4ECYP1A2CYP3A4
SCHEMBL8948062 0.74 HTR1A (0.69) HTR1ASIGMAR1HTR2C
SCHEMBL8948135 0.74 HTR2A (0.57) HTR2ASLC6A4SLC6A3HTR1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed