SCHEMBL8948117

SCHEMBL8948117

Cn1c(=O)oc2cc(C(=O)CBr)ccc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.62
HPGD P15428 1/20 0.62
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
SIGMAR1 Q99720 2/20 0.48
POLB P06746 2/20 0.48
TP53 P04637 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TSHR P16473 2/20 0.46
LMNA P02545 2/20 0.46
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GSK3B P49841 1/20 0.43
PKM P14618 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CBX7 O95931 1/20 0.43
CDYL Q9Y232 1/20 0.43
CDY1; CDY1B Q9Y6F8 1/20 0.43
GFER P55789 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10393870 0.89 ALDH1A1 (0.59) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL19513025 0.88 ALDH1A1 (0.51) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL10392904 0.87 ALDH1A1 (0.63) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL8787295 0.86 ALDH1A1 (0.56) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL14741026 0.84 ALDH1A1 (0.60) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL9684618 0.83 ALDH1A1 (0.63) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL8541265 0.83 ALDH1A1 (0.59) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL9367537 0.82 ALDH1A1 (0.58) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL5171751 0.81 ALDH1A1 (0.68) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL474056 0.81 ALDH1A1 (0.73) ALDH1A1HPGDKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed
US-4558060-A HYPNOTIC PROPERTIES; ANTI-HEART FAILURE MEDICINE RIOM LABORATORIES - CERM S.A. (FR) 1985-12-10 US disclosed