SCHEMBL8949066

SCHEMBL8949066

CCOC(=O)CCNC(=O)c1cc(-c2ccc(C#N)cc2)nn(C)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
TNF P01375 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
MAPK1 P28482 1/20 0.42
EGLN1 Q9GZT9 5/20 0.41
LMNA P02545 2/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
RAB9A P51151 1/20 0.40
PHGDH O43175 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
CHRM4 P08173 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
CASP1 P29466 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SLC34A1 Q06495 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9264740 0.95 ALDH1A1 (0.42) ALDH1A1KDM4EGAAHPGDTNF
Hydrochloric Acid SCHEMBL8949308 0.87 KDM1A (0.40) ALDH1A1KDM4EGAAHPGDTNF
SCHEMBL9571680 0.85 EGLN1 (0.42) ALDH1A1KDM4EGAAHPGDEGLN1
SCHEMBL7276252 0.82 HPGD (0.57) ALDH1A1KDM4EGAAHPGDMAPK1
SCHEMBL8949190 0.82 PHGDH (0.43) ALDH1A1KDM4EGAAHPGDMAPK1
SCHEMBL8410208 0.76 MAPT (0.52) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL7275259 0.75 PHGDH (0.48) ALDH1A1KDM4EGAAHPGDPHGDH
SCHEMBL8949139 0.74 KDM5B (0.39) HPGDPHGDHSMN1; SMN2
SCHEMBL8949288 0.74 KDM4E (0.43) ALDH1A1KDM4EGAAHPGDLMNA
SCHEMBL3929566 0.74 MAPT (0.55) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed