SCHEMBL8949190

SCHEMBL8949190

Cn1nc(-c2ccc(C#N)cc2)cc(C(=O)NCCCCC(=O)O)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.43
HDAC3 O15379 5/20 0.43
HDAC4 P56524 5/20 0.43
HDAC1 Q13547 5/20 0.43
HDAC2 Q92769 5/20 0.43
HDAC8 Q9BY41 5/20 0.43
HDAC6 Q9UBN7 5/20 0.43
HDAC7 Q8WUI4 4/20 0.43
HDAC10 Q969S8 4/20 0.43
HDAC11 Q96DB2 4/20 0.43
HDAC9 Q9UKV0 4/20 0.43
HDAC5 Q9UQL6 4/20 0.43
EGLN1 Q9GZT9 7/20 0.41
CHRM4 P08173 1/20 0.40
AOC3 Q16853 1/20 0.40
EGLN2 Q96KS0 2/20 0.39
MAPK1 P28482 1/20 0.38
KDM1A O60341 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9571680 0.87 EGLN1 (0.42) PHGDHHDAC3HDAC4HDAC1HDAC2
SCHEMBL8949033 0.83 ITGB3 (0.51) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL8949066 0.82 ALDH1A1 (0.46) PHGDHEGLN1CHRM4MAPK1KDM4E
SCHEMBL8949063 0.80 ITGB3 (0.47) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL5230660 0.80 HDAC3 (0.44) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL7275259 0.79 PHGDH (0.48) PHGDHEGLN2KDM4EALDH1A1GAA
Hydrochloric Acid SCHEMBL8949308 0.78 KDM1A (0.40) PHGDHEGLN1AOC3MAPK1KDM1A
Hydrochloric Acid SCHEMBL9264740 0.78 ALDH1A1 (0.42) PHGDHEGLN1CHRM4MAPK1KDM1A
SCHEMBL8949239 0.76 ITGB3 (0.45)
SCHEMBL8949269 0.75 EGLN1 (0.47) PHGDHEGLN1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed