SCHEMBL8949342

SCHEMBL8949342

CCOC(=O)c1ncn(CC(C(N)=O)C(C)(C)c2ccc(Cl)cc2)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.44
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.37
CYP19A1 P11511 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
TARBP2 Q15633 1/20 0.37
GABRG2 P18507 3/20 0.37
GABRB3 P28472 3/20 0.37
GABRA5 P31644 3/20 0.37
ELANE P08246 1/20 0.36
GABRA2 P47869 3/20 0.36
GABRB2 P47870 3/20 0.36
GABRA1 P14867 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA4 P48169 1/20 0.36
GABRA6 Q16445 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949213 0.86 SMN1; SMN2 (0.39) SCDNPC1RAB9AKDM4EMAPT
SCHEMBL8949336 0.73 KDM4E (0.41) SCDNPC1RAB9AKDM4EMAPT
SCHEMBL4958152 0.67 TSHR (0.54) SCDNPC1RAB9AKDM4ECYP19A1
SCHEMBL18764736 0.66 ALDH1A1 (0.42) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL10566878 0.66 ALDH1A1 (0.52) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL1903612 0.65 CYP3A4 (0.50) MAPTSMN1; SMN2LMNAPOLBGRIN2D
SCHEMBL28679512 0.65 GABRA2 (0.55) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL12604388 0.64 SCD (0.74) SCDKDM4EMAPTSMN1; SMN2MAPK1
SCHEMBL5990662 0.64 ALDH1A1 (0.47) KDM4EMAPTGABRG2GABRB3GABRA5
SCHEMBL30739186 0.63 SMN1; SMN2 (0.39) SCDCYP19A1SMN1; SMN2GABRA5GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547972-A 1-(ARLALKYLAMINOALKYL) IMIDAZOLE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1996-08-20 US disclosed
EP-0618907-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS Knoll AG (DE) 1994-10-12 EP disclosed
WO-1993013075-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed