SCHEMBL8949422

SCHEMBL8949422

N=C(N)c1ccc(-c2cc(C(=O)N[C@H]3CC[C@H](C(=O)O)CC3)c(N3CCCCC3)nn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
ITGB3 P05106 3/20 0.41
ITGA2B P08514 3/20 0.41
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
ACVR1 Q04771 1/20 0.40
F2 P00734 8/20 0.40
ST14 Q9Y5Y6 7/20 0.40
PRSS1 P07477 6/20 0.40
PRSS2 P07478 6/20 0.40
PRSS3 P35030 6/20 0.40
PLG P00747 2/20 0.40
MAPK13 O15264 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949409 0.99 ITGB3 (0.41) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8949406 0.91 MAPK14 (0.43) ITGB3ITGA2BBMPR1BBMPR1ATGFBR1
SCHEMBL8949300 0.91 ITGB3 (0.39) ITGB3ITGA2BF2ST14PRSS1
Hydrochloric Acid SCHEMBL8949012 0.90 MAPK13 (0.40) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8949089 0.90 ITGB3 (0.40) ITGB3ITGA2BBMPR1BBMPR1ATGFBR1
Hydrochloric Acid SCHEMBL8949020 0.89 TMPRSS15 (0.39) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL8949212 0.81 TMPRSS15 (0.40) ITGB3ITGA2BF2ST14PRSS1
Hydrochloric Acid SCHEMBL8949417 0.81 MAPK14 (0.42) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
Hydrochloric Acid SCHEMBL8949151 0.81 TMPRSS15 (0.37) ITGB3ITGA2BBMPR1BBMPR1AACVRL1
SCHEMBL8949341 0.80 KLK7 (0.45) MEN1KMT2AITGB3ITGA2BBMPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed