SCHEMBL8949995

SCHEMBL8949995

Cc1nc(C)c(C=O)c(-c2ccc(F)cc2)c1C=O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
PTGS2 P35354 6/20 0.42
AR P10275 4/20 0.42
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GCGR P47871 2/20 0.38
BRD4 O60885 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CASP3 P42574 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960475 0.87 MEN1 (0.43) ALDH1A1PTGS2ARMEN1KMT2A
SCHEMBL8949673 0.86 GCGR (0.50) ALDH1A1GCGR
SCHEMBL8949833 0.84 PTGS2 (0.38) ALDH1A1PTGS2ARMEN1KMT2A
SCHEMBL6955874 0.80 GCGR (0.61) ARGCGR
SCHEMBL7557484 0.77 EGLN1 (0.40) ALDH1A1PTGS2KMT2A
SCHEMBL8949603 0.77 GCGR (0.58) GCGR
SCHEMBL10656381 0.77 FABP3 (0.50) KDM4ELMNACASP3SMN1; SMN2
SCHEMBL9872802 0.76 GCGR (0.45) GCGR
SCHEMBL6956685 0.76 HMGCR (0.51) ALDH1A1PTGS2MEN1KMT2ANPC1
SCHEMBL9264457 0.74 MEN1 (0.41) ALDH1A1PTGS2ARMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502057-A Polysubstituted pyridines useful for treating lipoproteinanaemia and arteriosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1996-03-26 US disclosed
US-5470982-A Disubstituted pyridines BAYER AKTIENGESELLSCHAFT (DE) 1995-11-28 US disclosed
EP-0325129-B1 Disubstituted pyridines BAYER AG (DE) 1994-09-07 EP disclosed
US-5173495-A 7-[(2,6-dialkyl-4-furyl or thienyl-pyridyl)]-3,5-di-(dihydroxy-6-enoates) useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1992-12-22 US disclosed
US-4968689-A Certain 2,6-diisopropyl-4-(4-fluoro-phenyl)-3,5-bis-dimethyl-3',5'-dihydroxy-hept-6-enoate-pyridine derivatives useful for treating lipoproteinaemia and arteriosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed
EP-0325129-A2 Disubstituted pyridines BAYER AG (DE) 1989-07-26 EP disclosed