SCHEMBL8950322

SCHEMBL8950322

CC(C)n1ncnc1-c1ccc(CN)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
ADRB2 P07550 1/20 0.40
BPTF Q12830 1/20 0.39
AKT2 P31751 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
PIK3CA P42336 6/20 0.35
PIK3CB P42338 4/20 0.35
PIK3CD O00329 3/20 0.35
PIK3CG P48736 3/20 0.35
F9 P00740 1/20 0.35
F11 P03951 1/20 0.35
F7 P08709 1/20 0.35
CYP2C9 P11712 1/20 0.35
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
HCK P08631 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950355 0.81 HRH3 (0.47) DGAT1HRH3TAAR1ADRA1DADRA1A
SCHEMBL24185681 0.78 DGAT1 (0.41) DGAT1ADRA1DADRA1APIK3CAPIK3CB
SCHEMBL8997484 0.78 HRH3 (0.45) HRH3ADRB2BPTFAKT2LOXL2
SCHEMBL8950122 0.76 TDP1 (0.42) DGAT1ADRA1DADRA1APIK3CAPIK3CB
SCHEMBL31625362 0.70 AOC3 (0.39) HRH3ADRB2BPTFAKT2TAAR1
SCHEMBL17768600 0.70 BPTF (0.31) BPTF
SCHEMBL8950490 0.69 ADRA1D (0.36) DGAT1ADRA1DADRA1APIK3CAPIK3CB
SCHEMBL8950114 0.69 ADRA1D (0.36) DGAT1ADRA1DADRA1APIK3CAPIK3CB
SCHEMBL8950433 0.66 KDR (0.53) DGAT1PIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL25975917 0.65 SYK (0.42) HRH3ADRB2AKT2LOXL2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 DGAT1 842/4885HRH3 2616/4885ADRB2 4592/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.