SCHEMBL8950386

SCHEMBL8950386

CCOC(=O)CN(C)S(=O)(=O)c1ccsc1C1OCCO1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 2/20 0.37
ADRB2 P07550 1/20 0.36
ALOX15 P16050 1/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 2/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950198 0.82 GAA (0.36) GAAALDH1A1TSHRADRB2ALOX15
SCHEMBL11478128 0.75 ALDH1A1 (0.50) GAAALDH1A1MAPTPOLBKMT2A
SCHEMBL8950311 0.72 ALDH1A1 (0.34) GAAALDH1A1TSHRKDM4EMAPT
SCHEMBL7117736 0.71 GAA (0.49) GAAALDH1A1TSHRKDM4EMAPT
SCHEMBL8950073 0.66 ALDH1A1 (0.55) GAAALDH1A1MAPTLMNA
SCHEMBL11482764 0.66 KMT2A (0.53) GAAALDH1A1ADRB2ALOX15MAPT
SCHEMBL7673729 0.66 ALDH1A1 (0.56) GAAALDH1A1ADRB2ALOX15KDM4E
SCHEMBL8862623 0.65 ALDH1A1 (0.43) ALDH1A1TSHRKDM4ECYP3A4CYP2C9
SCHEMBL6501728 0.65 KMT2A (0.59) GAAALDH1A1TSHRADRB2ALOX15
SCHEMBL2332913 0.64 ADRB2 (0.65) GAAALDH1A1TSHRADRB2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022099-A1 OPHTHALMIC COMPOSITIONS FOR TREATING GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-25 WO disclosed
US-5538966-A ENZYME INHIBITORS FOR TREATMENT OF GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-23 US disclosed
WO-1995019981-A1 THIENOTHIAZINE SULFONAMIDE DERIVATIVES PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS CARBONIC ANHYDRASE INHIBITORS ALCON LABORATORIES, INC. (US) 1995-07-27 WO disclosed