SCHEMBL8952292

SCHEMBL8952292

O=C1NC(=O)C(OCc2ccccc2)C(=O)N1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
MMP2 P08253 2/20 0.42
MMP13 P45452 1/20 0.42
PDPK1 O15530 1/20 0.41
MTOR P42345 1/20 0.41
PPARG P37231 1/20 0.41
PSEN1 P49768 4/20 0.41
PSEN2 P49810 4/20 0.41
APH1B Q8WW43 4/20 0.41
NCSTN Q92542 4/20 0.41
APH1A Q96BI3 4/20 0.41
PSENEN Q9NZ42 4/20 0.41
ALDH1A1 P00352 4/20 0.40
TSHR P16473 1/20 0.40
MAPT P10636 1/20 0.40
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
CTSV O60911 1/20 0.39
CTSL P07711 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10411048 0.73 PDPK1 (0.35) BCHEACHEPDPK1MTORPSEN1
SCHEMBL5836429 0.73 ALDH1A1 (0.48) BCHEACHEMMP2MMP13PPARG
SCHEMBL29289313 0.71 ALDH1A1 (0.44) BCHEACHEPDPK1MTORPSEN1
SCHEMBL12597095 0.71 BCHE (0.42) BCHEACHEPDPK1MTORPSEN1
SCHEMBL320007 0.71 HSD17B10 (0.53) ALDH1A1MAPTMAOB
SCHEMBL3173157 0.71 BCHE (0.41) BCHEACHEPSEN1PSEN2APH1B
SCHEMBL2930554 0.70 SLC6A2 (0.54) MMP2MMP13PPARGALDH1A1TSHR
SCHEMBL21597997 0.70 GLA (0.56) ALDH1A1
SCHEMBL31579542 0.70 MMP13 (0.56) MMP2MMP13PPARGMAPTMAOA
SCHEMBL1929688 0.70 CRBN (0.44) BCHEACHEPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0725641-A4 1996-09-04 EP claimed
EP-0725641-A1 NOVEL ENZYME INHIBITORS, THEIR SYNTHESIS, AND METHODS FOR USE El Kouni, Mahmoud H. (US) 1996-08-14 EP claimed
WO-1995012400-A1 NOVEL ENZYME INHIBITORS, THEIR SYNTHESIS, AND METHODS FOR USE UAB RESEARCH FOUNDATION (US) 1995-05-11 WO claimed