SCHEMBL8955239

SCHEMBL8955239

O=C(Cc1ccc(Cl)c(Cl)c1)N1CCCC2CCC(N3CCCC3)C21

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 13/20 0.69
OPRM1 P35372 5/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9743230 0.99 OPRK1 (0.67) OPRK1OPRM1
SCHEMBL9669600 0.97 OPRK1 (0.73) OPRK1OPRM1
SCHEMBL9788886 0.97 OPRK1 (0.73) OPRK1OPRM1
SCHEMBL9669595 0.97 OPRK1 (0.73) OPRK1OPRM1
SCHEMBL9672001 0.96 OPRK1 (0.72) OPRK1OPRM1
Hydrochloric Acid SCHEMBL9742939 0.96 OPRK1 (0.69) OPRK1OPRM1
SCHEMBL9669607 0.83 OPRM1 (0.59) OPRK1OPRM1
SCHEMBL16237575 0.82 OPRK1 (0.82) OPRK1OPRM1
SCHEMBL17768434 0.82 OPRK1 (0.82) OPRK1OPRM1
SCHEMBL3765258 0.81 OPRK1 (1.00) OPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306356-B1 CONDENSED PIPERIDINE DERIVATIVES, INTERMEDIATES AND PROCESS FOR THEIR PREPARATION , THEIR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-05-19 EP claimed
US-5126353-A Also used as analgesics, diuretics, hypotensive agents, antiischemic agents ROUSSEL UCLAF (FR) 1992-06-30 US claimed
US-4927832-A DIURETIC, ANTIARRYTHMIA, ANTIISCHEMIC, HYPOTENSIVE ROUSSEL UCLAF (FR) 1990-05-22 US claimed
EP-0306356-A1 Condensed piperidine derivatives, intermediates and process for their preparation , their use as medicaments and pharmaceutical compositions containing them ROUSSEL-UCLAF (FR) 1989-03-08 EP claimed
EP-0456279-B1 Condensed piperidine derivatives, intermediates and process for their preparation, their use as medicaments and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1996-01-03 EP disclosed
EP-0306356-B1 CONDENSED PIPERIDINE DERIVATIVES, INTERMEDIATES AND PROCESS FOR THEIR PREPARATION , THEIR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-05-19 EP disclosed
US-5126353-A Also used as analgesics, diuretics, hypotensive agents, antiischemic agents ROUSSEL UCLAF (FR) 1992-06-30 US disclosed
EP-0456279-A1 Condensed piperidine derivatives, intermediates and process for their preparation, their use as medicaments and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1991-11-13 EP disclosed
US-4927832-A DIURETIC, ANTIARRYTHMIA, ANTIISCHEMIC, HYPOTENSIVE ROUSSEL UCLAF (FR) 1990-05-22 US disclosed
EP-0306356-A1 Condensed piperidine derivatives, intermediates and process for their preparation , their use as medicaments and pharmaceutical compositions containing them ROUSSEL-UCLAF (FR) 1989-03-08 EP disclosed