SCHEMBL8957016

SCHEMBL8957016

COc1ccc2[nH]cc(CC(=O)N3C[C@@H]4[C@H](C3)C(c3ccccc3)(c3ccccc3)CC[C@@]4(O)c3ccccc3OC)c2c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.54
DRD2 P14416 5/20 0.49
DRD3 P35462 5/20 0.49
OPRK1 P41145 1/20 0.49
FNTA P49354 3/20 0.47
FNTB P49356 3/20 0.47
KDM4E B2RXH2 1/20 0.46
SIGMAR1 Q99720 1/20 0.44
ICMT O60725 1/20 0.43
DRD4 P21917 4/20 0.42
CXCR3 P49682 1/20 0.40
FAAH O00519 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9245521 1.00 TACR1 (0.54) TACR1DRD2DRD3OPRK1FNTA
SCHEMBL9243104 0.93 TACR1 (0.55) TACR1DRD2DRD3OPRK1FNTA
SCHEMBL8956827 0.93 TACR1 (0.55) TACR1DRD2DRD3OPRK1FNTA
SCHEMBL8956847 0.91 TACR1 (0.58) TACR1DRD2DRD3OPRK1FNTA
SCHEMBL8956681 0.91 TACR1 (0.58) TACR1DRD2DRD3OPRK1FNTA
SCHEMBL8893638 0.88 DRD2 (0.46) TACR1DRD2DRD3OPRK1FNTA
SCHEMBL8956909 0.83 TACR1 (0.67) TACR1FNTAFNTBKDM4ESIGMAR1
SCHEMBL8545840 0.83 TACR1 (0.67) TACR1FNTAFNTBKDM4ESIGMAR1
SCHEMBL9247977 0.82 TACR1 (0.64) TACR1FNTAFNTBSIGMAR1MEN1
SCHEMBL8956812 0.82 TACR1 (0.64) TACR1FNTAFNTBSIGMAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5484804-A Perhydroisoindole derivatives as antagonists of substance P RHONE-POULENC RORER S.A. (FR) 1996-01-16 US disclosed